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Umeå universitet
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Personalbild Pardeep Singh

Pardeep Singh

Kontakt

E-post
pardeep.singh@umu.se
Telefon
090-786 92 83

Verksam vid

Anknytning
Staff scientist vid Kemiska institutionen
Plats
KB.C4, Linnaeus väg 10, C4-39-07 Umeå universitet, 901 87 Umeå
Photoredox-catalyzed radical coupling of C7-chloromethyl-substituted thiazolino ring-fused 2-pyridones with quinoxalinones
Journal of Organic Chemistry, American Chemical Society (ACS) 2024, Vol. 89, (16) : 11802-11810
Hellgren, Victor; Singh, Pardeep; Kulkarni, Abhilash; et al.
Synthesis of three-dimensional ring fused heterocycles by a selective [4 + 2] cycloaddition between bicyclic thiazolo 2-pyridones and arynes
Journal of Organic Chemistry, American Chemical Society (ACS) 2024, Vol. 89, (1) : 731-739
Sarkar, Souvik; Singh, Pardeep; Edin, Simon; et al.
Dihydrothiazolo ring-fused 2-pyridone antimicrobial compounds treat Streptococcus pyogenes skin and soft tissue infection
Science Advances, American Association for the Advancement of Science (AAAS) 2024, Vol. 10, (31)
Zou, Zongsen; Singh, Pardeep; Pinkner, Jerome S.; et al.
A highly substituted ring-fused 2-pyridone compound targeting PrfA and the efflux regulator BrtA in listeria monocytogenes
mBio, American Society for Microbiology 2023, Vol. 14, (3)
Tükenmez, Hasan; Singh, Pardeep; Sarkar, Souvik; et al.
Ring-fused 2-pyridones effective against multidrug-resistant Gram-positive pathogens and synergistic with standard-of-care antibiotics
Proceedings of the National Academy of Sciences of the United States of America, PNAS 2022, Vol. 119, (43)
Nye, Taylor M.; Tükenmez, Hasan; Singh, Pardeep; et al.
K2S2O8-mediated coupling of 6-amino-7-aminomethyl-thiazolino-pyridones with aldehydes to construct amyloid affecting pyrimidine-fused thiazolino-2-pyridones
Organic and biomolecular chemistry, The Royal Society of Chemistry 2021, Vol. 19, (44) : 9758-9772
Bharate, Jaideep B.; Ådén, Jörgen; Gharibyan, Anna; et al.
An efficient and scalable synthesis of thiazolo ring fused 2-pyridones using flow chemistry
ARKIVOC, Arkat 2021, Vol. 2020, (7) : 365-378
Cairns, Andrew G.; Sarkar, Souvik; Singh, Pardeep; et al.
A 2-pyridone amide inhibitor of transcriptional activity in Chlamydia trachomatis
Antimicrobial Agents and Chemotherapy, American Society for Microbiology 2021, Vol. 65, (5)
Núñez-Otero, Carlos; Bahnan, Wael; Vielfort, Katarina; et al.
Tandem Ring Opening/Intramolecular [2 + 2] Cycloaddition Reaction for the Synthesis of Cyclobutane Fused Thiazolino-2-Pyridones
Journal of Organic Chemistry, American Chemical Society (ACS) 2021, Vol. 86, (23) : 16582-16592
Tyagi, Mohit; Adolfsson, Dan E.; Singh, Pardeep; et al.
Intramolecular Povarov Reactions for the Synthesis of Chromenopyridine fused 2-Pyridone Polyheterocycles Binding to α-Synuclein and Amyloid-β fibrils
Journal of Organic Chemistry, American Chemical Society (ACS) 2020, Vol. 85, (21) : 14174-14189
Adolfsson, Dan E.; Tyagi, Mohit; Singh, Pardeep; et al.
Methyl sulfonamide substituents improve the pharmacokinetic properties of bicyclic 2-pyridone based Chlamydia trachomatis inhibitors
MedChemComm, Royal Society of Chemistry 2019, Vol. 10, (11) : 1966-1987
Kulén, Martina; Núñez-Otero, Carlos; Cairns, Andrew G.; et al.
Visible light mediated synthesis of β chloro ketones from aryl cyclopropanes
Angewandte Chemie International Edition, John Wiley & Sons 2019, Vol. 58 : 8577-8580
Petzold, Daniel; Singh, Pardeep; Almqvist, Fredrik; et al.
Pyridine-Fused 2-Pyridones via Povarov and A3 Reactions: Rapid Generation of Highly Functionalized Tricyclic Heterocycles Capable of Amyloid Fibril Binding
Journal of Organic Chemistry, American Chemical Society (ACS) 2019, Vol. 84, (7) : 3887-3903
Singh, Pardeep; Adolfsson, Dan E.; Ådén, Jörgen; et al.
Synthesis of Densely Functionalized N-Alkenyl 2-Pyridones via Benzyne-Induced Ring Opening of Thiazolino-Fused 2-Pyridones
Organic Letters, American Chemical Society (ACS) 2019, Vol. 21 : 6946-6950
Singh, Pardeep; Cairns, Andrew G.; Adolfsson, Dan E.; et al.
β‐Lactam‐Synthon Interceded Diastereoselective Synthesis of 2‐Azido‐γ‐amino Alcohols with Subsequent Transformations to Functionally Enriched Heterocycles
ChemistrySelect, John Wiley & Sons 2018, Vol. 3, (17) : 4764-4767
Singh, Amandeep; Sharma, Bharvi; Sachdeva, Divya; et al.
Synthesis of multiring fused 2‑pyridones via a nitrene insertion reaction: fluorescent modulators of α‑synuclein amyloid formation
Organic Letters, American Chemical Society (ACS) 2015, Vol. 17, (24) : 6194-6197
Singh, Pardeep; Chorell, Erik; Krishnan, K Syam; et al.
Enhanement of amyloid fibril binding by ring expansion of thiazolino fused 2-pyridone peptidomimetics
Adolfsson, Dan E.; Tyagi, Mohit; Singh, Pardeep; et al.
K2S2O8-mediated aerobic oxidative coupling of 6-amino-7-(aminomethyl)-thiazolino-pyridones with aldehydes: Direct access to highly functionalized pyrimidine fused thiazolino-2-pyridones with amyloid fibril binding activity or inhibitors of Amyloid-β fibril formation
Bharate, Jaideep B.; Ådén, Jörgen; Gharibyan, Anna; et al.
Discovery of three new binding sites and modes of ring-fused 2-pyridones to PrfA: How can they contribute to drug design?
Oelker, Melanie; Vielfort, Katarina; Lindgren, Cecilia; et al.
Functionalization of Thiazolino fused 2-Pyridones by thiazoline ring opening and closing: Identification of new Amyloid Binding Heterocycles
Tyagi, Mohit; Adolfsson, Dan E.; Ådén, Jörgen; et al.
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